Showing 13–20 of 20 results
|CAS NO.||PRODUCT NAME||OVERVIEW|
|656247-17-5||Nintedanib (BIBF 1120) (656247-17-5)||
Nintedanib(BIBF 1120) is a member of the class of oxindoles that is a kinase inhibitor used (in the form of its ethylsulfonate salt) for the ...
PD173074 is a member of the class of ureas that is 1-tert-butylurea in which one of the hydrogens attached to N(3) is substituted by a pyrido...
SKLB610 is a VEGFR inhibitor that potently suppresses human tumor angiogenesis. SKLB610 exhibited its antitumor activity as a multi-targeted...
SSR128129E (SSR) is an potent FGFR inhibitor, which inhibits fibroblast growth factor receptor (FGFR) signaling by binding to the extracellul...
|341031-54-7||Sunitinib Malate (341031-54-7)||
Sunitinib Malate is the orally bioavailable malate salt of an indolinone-based tyrosine kinase inhibitor with potential antineoplastic activi...
|905854-02-6||Tivantinib (ARQ197) (905854-02-6)||
Tivantinib (ARQ197) has been shown to prevent HGF/c-met induced cellular responses in vitro. Tivantinib (ARQ197) possesses antitumor activity...
|475108-18-0||Tivozanib (AV-951) (475108-18-0)||
Tivozanib (AV-951) is a potent and selective VEGFR inhibitor for VEGFR1/2/3 with IC50 of 30 nM/6.5 nM/15 nM, and also inhibits PDGFR and c-Ki...
|252916-29-3||TSU-68 (SU6668) (252916-29-3)||
TSU-68(SU6668,Orantinib) has greatest potency against PDGFR autophosphorylation with Ki of 8 nM in a cell-free assay, but also strongly inhib...
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