Showing 1–12 of 13 results
|CAS NO.||PRODUCT NAME||OVERVIEW|
|30827-99-7||AEBSF HCL (30827-99-7)||
AEBSF or 4-(2-aminoethyl)benzenesulfonyl fluoride hydrochloride is a water-soluble, irreversible serine protease inhibitor with a molecular w...
AMG-3969 is a potent, metabolically stable Glucokinase (GK)-GKRP (GK regulatory protein) disruptor with IC50 of 4 nM, does not block the GK b...
AP-III-a4 (ENOblock) is the first nonsubstrate analogue inhibitor of enolase with IC50 of 0.576 μM.
BMS-378806 selectively inhibits the binding of HIV-1 gp120 to the CD4 receptor with EC50 of 0.85-26.5 nM in virus.
E-6005, also known as RVT-501 and lotamilast, is a phosphodiesterase 4 (PDE-4) inhibitor potentially for the treatment of atopic dermatitis.<...
LCI699, also known as Osilodrostat, is a potent inhibitor of 11β-hydroxylase, the enzyme which catalyzes the final step of cortisol synthesis...
|173039-10-6||PMPA (NAALADaseinhibitor) (173039-10-6)||
PMPA is a selective inhibitor of NAALADase with Ki value of 275 pM.PMPA is a potent NAALADase inhibitor and has a more activity than reported...
TMS5275 is an orally available, potent and selective inhibitor of PAI-1 that delivers antithrombotic benefits devoid of bleeding effect in no...
TM5441 is a plasminogen activator inhibitor-1 (PAI-1); inhibits several tumor cell lines with IC50 values between 9.7 and 60.3 μM.
Vadadustat is a novel, titratable, oral hypoxia-inducible factor prolyl hydroxylase (HIF-PH) inhibitor in development for the treatment of an...
XMD16-5 is a novel tyrosine kinase nonreceptor 2(TNK2) inhibitor with IC50s of 16 nmol/L and 77 nmol/L for the D163E and R806Q mutations....
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