Showing 1–12 of 53 results
|CAS NO.||PRODUCT NAME||OVERVIEW|
Iodopravadoline, also known as AM630, is an inverse agonist at the human cannabinoid CB1 receptor. Iodopravadoline has been found to attenuat...
Amiselimod hydrochloride is a novel sphingosine 1-phosphate receptor-1 (S1P1) modulator, designed to reduce the bradycardia effects associate...
APD334, also known as Etrasimod, is a potent, centrally available, functional antagonists of the S1P1 receptor for use as next generation the...
ARS-853 (ARS853) is a selective, covalent KRAS(G12C) inhibitor that inhibits mutant KRAS-driven signaling by binding to the GDP-bound oncopro...
Bay 59-3074 is a novel, selective CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors respecti...
BIBS39 is a nonpeptide angiotensin II (AII) receptor antagonists that displaced [125I] AII from its specific binding sites with a K(i) value ...
BLU-285 is a dual inhibitor of KIT receptor and platelet-derived growth factor receptor α (PDGFRα) tyrosine kinases with activating loop muta...
BMS-986020, is a potent G protein-coupled lysophosphatidic acid receptor 1 (LPA1) antagonist. BMS-986020 , also known as AM152 and AP-3152 fr...
BQU57, a derivative of RBC8, is a selective GTPase Ral inhibitor relative to the GTPases Ras and RhoA.
CEP-40783, also known as RXDX-106,is an orally-available, potent and selective TAM(TYRO3, AXL, MER)/MET inhibitor displaying low nanomolar bi...
|124431-80-7||CGS21680 HCL (124431-80-7)||
CGS 21680 HCL is a potent, selective agonist of the adenosine A2A receptor (Ki = 11-46 nM).It is less effective at adenosine A1 and A3 recept...
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