Showing 1–12 of 20 results
|CAS NO.||PRODUCT NAME||OVERVIEW|
BIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 μM. BIX01294 is an inhibitor of G9a histone methyltransferase with...
BMH-21 is a small molecule DNA intercalator that binds ribosomal DNA and inhibits RNA polymerase I (Pol I) transcription; does not cause phos...
|168425-64-7||Compound 401 (168425-64-7)||
Compound 401 is a synthetic inhibitor of DNA-PK (IC50 = 0.28 μM) that also targets mTOR but not PI3K.Compound 401 is a cell-permeable pyrimid...
CRT0044876 is a potent and selective APE1 inhibitor with IC50 of ~3 μM. CRT0044876 is a potent and selective APE1 inhibitor. In HeLa whole ce...
CX-5461 is an inhibitor of rRNA synthesis, selectively inhibits Pol I-driven transcription of rRNA with IC50 of 142 nM, has no effect on Pol ...
|259793-96-9||Favipiravir (T-705) (259793-96-9)||
Favipiravir (T-705) is a potent and selective RNA-dependent RNA polymerase inhibitor, used to treat influenza virus infections. Favipiravir, ...
GSK126 is an effective EZH2 methyltransferase inhibitor with IC50 being 9.9nM and high selectivity on EZH2 which is over 1000 times higher th...
|57852-57-0||Idarubicin HCl (57852-57-0)||
Idarubicin HCl is a hydrochloride salt form of Idarubicin which is an anthracycline antibiotic and a DNA topoisomerase II (topo II) inhibitor...
Lomeguatrib is a O6-methylguanine-DNA methyltransferase (MGMT) inhibitor, with IC50s of 9 nM in cell-free assay and ∼6 nM in MCF-7 cells̷...
NMS-P715 is an orally bioavailable, ATP-competitive, reversible, and time-dependent inhibitor of MPS1 (IC50 = 182 nM, Ki = 0.99 nM)., The MPS...
NU7441 (KU-57788) is a highly potent and selective DNA-PK inhibitor with IC50 of 14 nM and also inhibits PI3K with IC50 of 5 μM….<...
Pirarubicin is an anthracycline antibiotic, and also a DNA/RNA synthesis inhibitor by intercalating into DNA and interacts with topoisomerase...
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