Showing 1–12 of 36 results
|CAS NO.||PRODUCT NAME||OVERVIEW|
(-)-Blebbistatin is a cell-permeable inhibitor for non muscle myosin II ATPase with IC50 of ~2 μM, does not inhibit myosin light chain kinase...
(+)-JQ1 is a BET bromodomain inhibitor, with IC50 of 77 nM/33 nM for BRD4(1/2),binding to all bromodomains of the BET family, but not to brom...
AMG 517 is a potent and selective TRPV1 antagonist, antagonizes capsaicin, proton, and heat activation of TRPV1 with IC50 of 0.76 nM, 0.62 nM...
Andarine is a selective non-steroidal androgen receptor (AR) agonist with Ki of 4 nM, tissue-selective for anabolic organs….
AZ20 is a novel potent and selective inhibitor of ATR kinase with IC50 of 5 nM, 8-fold selectivity over mTOR. AZ20 is an ATR protein kinase i...
AZD0156 is an oral, potent and selective ATM kinase inhibitor, inhibiting the kinase activity of ATM and ATM-mediated signaling, preventing D...
AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μMand has ability of reducing AR protein expression…
AZD4547 is a novel selective FGFR inhibitor targeting FGFR1/2/3 with IC50 of 0.2 nM/2.5 nM/1.8 nM, weaker activity against FGFR4, VEGFR2(KDR)...
AZD6738 is a potent selective oral ATR inhibitor. It can inhibit ATR substrate Chk1 Ser345 phosphorylation in cells with an IC50 value of 74 ...
AZD7762 is a potent and selective inhibitor of Chk1 with IC50 of 5 nM. It is equally potent against Chk2 and less potent against CAM, Yes, Fy...
|847499-27-8||CEP-18770 (Delanzomib) (847499-27-8)||
CEP-18770 is an orally active inhibitor of the chymotrypsin-like activity of proteasome with IC50 of 3.8 nM, with only marginal inhibition of...
CGK 733 is a potent and selective inhibitor of ATM/ATR with IC50 of ~200 nM. CGK733 is an ATM inhibitor and ATR inhibitor, which significantl...
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